Buprenorphine Formulations

In the US, there are several buprenorphine options, primarily categorized as buprenorphine monoproducts and buprenorphine-naloxone combination products. Here is a quick review of what is widely available at VA. Note that buprenorphine is also available in an IV formulation, but not widely available within VA (yet).

  • Suboxone (Buprenorphine/Naloxone Combination):

    • Administered sublingually or buccally (between the gum and cheek).

    • Combines buprenorphine with naloxone to deter intravenous misuse.

    • Available in both film and tablet forms.

  • Subutex (Buprenorphine Monotherapy):

    • Administered sublingually (under the tongue).

    • Typically used at the initiation of treatment.

    • Available in tablet form.

  • Belbuca (Buprenorphine Buccal Film):

    • Primarily indicated for chronic pain management.

    • Administered buccally.

    • Provides continuous pain relief with a lower risk of dependency.

  • Butrans (Buprenorphine Transdermal Patch):

    • Administered transdermally (through the skin).

    • Primarily indicated for chronic pain management.

    • Provides continuous pain relief for up to seven days.

    • Designed for patients requiring around-the-clock opioid treatment.

  • Sublocade (Buprenorphine Extended-Release Injection):

    • Administered subcutaneously (under the skin) once a month.

    • Provides long-acting effects and has been shown to maintain therapeutic levels of buprenorphine over a month.

  • Brixadi (Buprenorphine Extended-Release Injection):

    • Administered subcutaneously (under the skin) once a week or once a month.

    • Designed for the treatment of opioid use disorder.

    • Provides flexible dosing options to maintain therapeutic levels of buprenorphine.

  • Buprenex (Buprenorphine Injection):

    • Administered intravenously or intramuscularly.

    • Primarily used for the management of moderate to severe pain.

    • Provides rapid pain relief in a clinical setting.

Reference:

1.         Buprenorphine: Drug Information. UpToDate website. https://www.uptodate.com/contents/buprenorphine-drug-information?source=auto_suggest&selectedTitle=12---12---bupren&search=buprenorphine. Updated 2023. Accessed October 5, 2023.

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